SCHEMBL9433624

SCHEMBL9433624

COC(=O)C1=C(C)NC(C)=C(c2cccnc2)C1c1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 9/20 0.48
GAA P10253 4/20 0.46
HPGD P15428 4/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 4/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP3A4 P08684 1/20 0.44
KDM4E B2RXH2 4/20 0.43
HSD17B10 Q99714 4/20 0.43
CASP1 P29466 3/20 0.43
CASP7 P55210 3/20 0.43
SLC6A3 Q01959 1/20 0.43
GLA P06280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434358 0.92 GAA (0.46) GAAHPGDNPSR1ALDH1A1MAPK1
SCHEMBL10432258 0.90 GAA (0.48) GAAHPGDNPSR1ALDH1A1MAPK1
SCHEMBL9434716 0.89 CACNA1F (0.53) GAAHPGDNPSR1ALDH1A1SMN1; SMN2
SCHEMBL9434642 0.89 CACNA1B (0.52) CACNA1B
SCHEMBL10432716 0.88 CACNA1F (0.57) GAAHPGDNPSR1ALDH1A1CYP3A4
SCHEMBL9434208 0.88 GAA (0.46) CACNA1BGAAHPGDNPSR1ALDH1A1
SCHEMBL9434188 0.88 POLB (0.50) CACNA1BGAAHPGDNPSR1ALDH1A1
SCHEMBL10678279 0.87 CACNA1B (0.55) CACNA1BSLC6A3
SCHEMBL9434369 0.84 MAPT (0.63) MAPK1CYP3A4
SCHEMBL9434688 0.84 KDM4E (0.47) GAAHPGDNPSR1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed