SCHEMBL9434641

SCHEMBL9434641

CC(N)=CC(=O)OCC#Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
GAA P10253 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
THPO P40225 1/20 0.40
HTT P42858 1/20 0.39
SLC1A5 Q15758 2/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
ALOX5 P09917 1/20 0.39
HTR2A P28223 1/20 0.38
GRIK1 P39086 1/20 0.38
GRIK2 Q13002 1/20 0.38
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434629 1.00 CA12 (0.40) CA12CA1CA2CA7CA9
SCHEMBL9434020 0.90 GAA (0.35) CA12CA1CA2CA7CA9
SCHEMBL9434034 0.90 GAA (0.35) CA12CA1CA2CA7CA9
SCHEMBL7864231 0.84 CYP2A6 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19FFAR1
SCHEMBL7864229 0.84 CYP2A6 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19FFAR1
SCHEMBL27545848 0.79 ALDH1A1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL14784333 0.79 CYP1A2 (0.48) CA12CA1CA2CA7CA9
SCHEMBL9434090 0.79 PPARD (0.46) GAANPC1RAB9AFFAR1
SCHEMBL9434074 0.79 PPARD (0.46) GAANPC1RAB9AFFAR1
SCHEMBL25200657 0.76 GAA (0.44) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed