SCHEMBL7864229

SCHEMBL7864229

C/C(N)=C/C(=O)OCC#Cc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.48
CYP2C9 P11712 3/20 0.48
CYP2B6 P20813 3/20 0.48
CYP2C19 P33261 3/20 0.48
CYP2E1 P05181 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C8 P10632 1/20 0.47
CHRNB2 P17787 5/20 0.46
CHRNA4 P43681 5/20 0.46
FFAR1 O14842 1/20 0.40
GRM5 P41594 2/20 0.38
ERN1 O75460 1/20 0.38
PTAFR P25105 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TBXAS1 P24557 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864231 1.00 CYP2A6 (0.48) CYP2A6CYP2C9CYP2B6CYP2C19CYP2E1
SCHEMBL9434641 0.84 CA12 (0.40) CYP2C9CYP2C19CYP3A4CYP1A2FFAR1
SCHEMBL9434629 0.84 CA12 (0.40) CYP2C9CYP2C19CYP3A4CYP1A2FFAR1
SCHEMBL9434020 0.75 GAA (0.35) CYP2C9CYP2C19CYP3A4CYP1A2FFAR1
SCHEMBL9434034 0.75 GAA (0.35) CYP2C9CYP2C19CYP3A4CYP1A2FFAR1
SCHEMBL29883579 0.75 CYP19A1 (0.47) CYP2C9CYP3A4CYP1A2TBXAS1
SCHEMBL28764754 0.74 LMNA (0.52) CYP2A6CYP2C9CYP2B6CYP2C19CYP2E1
SCHEMBL8329404 0.73 CHRNA7 (0.54) CYP2A6PTAFRL3MBTL1TBXAS1
SCHEMBL8329403 0.73 CHRNA7 (0.54) CYP2A6PTAFRL3MBTL1TBXAS1
SCHEMBL7054843 0.72 CHRNB2 (0.55) CYP2A6CYP2C9CYP2B6CYP2C19CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed