SCHEMBL9434701

SCHEMBL9434701

C=CC(=O)Cc1cnccc1-c1cccc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.40
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
DAPK3 O43293 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CYP19A1 P11511 1/20 0.36
CDC7 O00311 1/20 0.36
MAPT P10636 1/20 0.36
TGM2 P21980 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP1A1 P04798 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP1B1 Q16678 1/20 0.36
IDO1 P14902 1/20 0.35
DGAT2 Q96PD7 2/20 0.35
KMT2A Q03164 2/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434756 0.86 CYP3A4 (0.39) CYP19A1CDC7CYP1A2CYP1A1CYP3A4
SCHEMBL9433871 0.85 PDE4A (0.37) CDC7MAPT
SCHEMBL9434449 0.85 RPS6KA3 (0.46) DAPK3KDM4ECDC7IDO1
SCHEMBL9434027 0.84 SLC22A12 (0.40) EGFRALDH1A1DAPK3KDM4ELMNA
SCHEMBL9434562 0.82 SLC22A12 (0.47) ALDH1A1CDC7CYP1A2CYP3A4CYP2D6
SCHEMBL9434742 0.82 GPBAR1 (0.41) CYP19A1CYP3A4DGAT2KMT2ACYP2C9
SCHEMBL9433930 0.81 GPBAR1 (0.36) ALDH1A1HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL9433405 0.81 PDE4A (0.43) ALDH1A1CDC7MAPTTGM2CYP1A2
SCHEMBL17520239 0.78 CCNC (0.48) ALDH1A1HPGDDAPK3KDM4ELMNA
SCHEMBL9433625 0.78 KMT2A (0.35) ALDH1A1HPGDKDM4ETGM2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed