SCHEMBL9433405

SCHEMBL9433405

C=CC(=O)Cc1cnccc1-c1cccc([N+](=O)[O-])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.43
PDE4C Q08493 2/20 0.43
PDE4D Q08499 2/20 0.43
PDE4B Q07343 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA4 P43681 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CDC7 O00311 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
TGM2 P21980 1/20 0.40
MAPT P10636 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433650 0.86 L3MBTL1 (0.40) POLBALDH1A1MEN1KMT2ATGM2
SCHEMBL9434756 0.82 CYP3A4 (0.39) CDC7CYP1A2CYP3A4CYP2C9
SCHEMBL9434449 0.81 RPS6KA3 (0.46) CDC7
SCHEMBL9434701 0.81 EGFR (0.40) SMN1; SMN2ALDH1A1MEN1KMT2ACDC7
SCHEMBL9433871 0.81 PDE4A (0.37) PDE4ACDC7MAPT
SCHEMBL9433812 0.79 MAPT (0.43) PDE4APDE4CPDE4DSMN1; SMN2ALDH1A1
SCHEMBL9434562 0.78 SLC22A12 (0.47) TDP1ALDH1A1CHRNB2CHRNA5CHRNA4
SCHEMBL9434742 0.78 GPBAR1 (0.41) PDE4ATDP1MEN1KMT2ACYP3A4
SCHEMBL9433598 0.78 RORC (0.40) TDP1SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL9433930 0.77 GPBAR1 (0.36) TDP1SMN1; SMN2ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3002161-A None JP disclosed
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
JP-H032161-A 1,4-DIHYDROPYRIDINE DERIVATIVE FUJIREBIO INC 1991-01-08 JP disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed