SCHEMBL9434879

SCHEMBL9434879

O=C1N(c2ccc(Cl)cc2)c2ncccc2C1(Cc1ccncc1)Cc1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
MAPK1 P28482 1/20 0.47
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
ALOX12 P18054 1/20 0.40
AOC2 O75106 1/20 0.40
KMT2A Q03164 1/20 0.39
PGR P06401 3/20 0.39
NAMPT P43490 3/20 0.39
ELANE P08246 2/20 0.38
ABCB1 P08183 1/20 0.38
DHODH Q02127 1/20 0.37
KCNQ2 O43526 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9304548 0.99 MAPK1 (0.49) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL9434703 0.93 ALDH1A1 (0.55) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL9302631 0.92 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL9303053 0.92 MAPK1 (0.55) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL9304013 0.86 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL9305548 0.85 MAPK1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL9211380 0.83 ALDH1A1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL9210703 0.82 MAPK1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
SCHEMBL9303463 0.81 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL9305520 0.81 MAPK1 (0.71) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994006793-A1 3,3'-DISUBSTITUTED-1,3-DIHYDRO-2H-PYRROLO[2,3-b]HETEROCYCLIC-2-ONE USEFUL IN THE TREATMENT OF COGNITIVE DISORDERS OF MAN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-03-31 WO claimed