SCHEMBL9435149

SCHEMBL9435149

O=C1CCc2c[c]cc(CCl)c2N1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
CRBN Q96SW2 1/20 0.32
BRD4 O60885 3/20 0.32
CYP1A2 P05177 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
CA9 Q16790 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434680 0.83 NPC1 (0.33) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL11266794 0.75 NPC1 (0.46) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL5546054 0.70 CYP11B1 (0.39) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL5542652 0.65 MAOB (0.51) CRBNBRD4CYP11B1CYP11B2
SCHEMBL17969062 0.62 NPC1 (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8919270 0.62 NPC1 (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL28628183 0.61 NPC1 (0.46) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2056143 0.61 BRD4 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL986343 0.61 NPC1 (0.55) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL7350316 0.60 NPC1 (0.41) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994025453-A1 4-ARYL-4-HYDROXY-TETRAHYDROPYRANS AND 3-ARYL-3-HYDROXY-TETRAHYDROFURANS AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-11-10 WO claimed
WO-1994025453-A1 4-ARYL-4-HYDROXY-TETRAHYDROPYRANS AND 3-ARYL-3-HYDROXY-TETRAHYDROFURANS AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-11-10 WO disclosed