SCHEMBL9435498

SCHEMBL9435498

COc1ccc(C2(C#N)CCC(N3CCN(CC(O)COc4ccc(F)cc4)CC3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
TSHR P16473 1/20 0.53
CACNA1G O43497 2/20 0.51
CYP2D6 P10635 5/20 0.49
KDM4E B2RXH2 2/20 0.48
POLB P06746 1/20 0.48
GLA P06280 1/20 0.46
DRD4 P21917 1/20 0.46
MAPT P10636 1/20 0.46
KCNH2 Q12809 1/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HTT P42858 1/20 0.45
RAD52 P43351 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435494 1.00 MEN1 (0.56) MEN1KMT2ATSHRCACNA1GCYP2D6
SCHEMBL9435568 0.95 TSHR (0.54) MEN1KMT2ATSHRCACNA1GKDM4E
SCHEMBL9435578 0.95 TSHR (0.54) MEN1KMT2ATSHRCACNA1GKDM4E
SCHEMBL9435774 0.92 TSHR (0.51) MEN1KMT2ATSHRCACNA1GKDM4E
SCHEMBL9435768 0.92 TSHR (0.51) MEN1KMT2ATSHRCACNA1GKDM4E
SCHEMBL9098349 0.91 TSHR (0.52) MEN1KMT2ATSHRCACNA1GCYP2D6
SCHEMBL9098357 0.91 TSHR (0.52) MEN1KMT2ATSHRCACNA1GCYP2D6
SCHEMBL9098366 0.91 TSHR (0.52) MEN1KMT2ATSHRCACNA1GCYP2D6
SCHEMBL9435813 0.91 CACNA1G (0.58) MEN1KMT2ATSHRCACNA1GCYP2D6
SCHEMBL9435818 0.91 CACNA1G (0.58) MEN1KMT2ATSHRCACNA1GCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371088-A 1-aryl-4-piperazinylcyclohexanecarbonitriles, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed