SCHEMBL9435568

SCHEMBL9435568

N#C[C@]1(c2ccc(F)cc2)CC[C@H](N2CCN(CC(O)COc3ccc(F)cc3)CC2)CC1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
CACNA1G O43497 9/20 0.49
KCNH2 Q12809 3/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
KDM4E B2RXH2 1/20 0.47
GLA P06280 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.46
RAD52 P43351 1/20 0.46
ABCB1 P08183 2/20 0.46
RRM1 P23921 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435578 1.00 TSHR (0.54) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9435774 0.96 TSHR (0.51) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9435768 0.96 TSHR (0.51) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9435498 0.95 MEN1 (0.56) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9435494 0.95 MEN1 (0.56) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9098357 0.95 TSHR (0.52) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9098349 0.95 TSHR (0.52) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9098366 0.95 TSHR (0.52) TSHRCACNA1GKCNH2MEN1KMT2A
SCHEMBL9435534 0.89 CACNA1G (0.57) TSHRCACNA1GKCNH2MAPT
SCHEMBL9435539 0.89 CACNA1G (0.57) TSHRCACNA1GKCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371088-A 1-aryl-4-piperazinylcyclohexanecarbonitriles, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed