SCHEMBL9436735

SCHEMBL9436735

COC(=O)c1ccc(Oc2ccccc2)c(S(N)(=O)=O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.56
KDM4E B2RXH2 3/20 0.51
HSD17B10 Q99714 2/20 0.51
P2RX4 Q99571 5/20 0.50
ALDH1A1 P00352 3/20 0.50
HPGD P15428 3/20 0.50
USP2 O75604 2/20 0.50
GAA P10253 1/20 0.50
F10 P00742 1/20 0.50
TTR P02766 2/20 0.49
CA2 P00918 3/20 0.49
CA1 P00915 2/20 0.49
CA9 Q16790 2/20 0.49
CA5A P35218 1/20 0.49
BRD4 O60885 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
ADRA2B P18089 1/20 0.46
HTR2C P28335 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230507 0.89 KDM4E (0.55) PKMKDM4EHSD17B10P2RX4ALDH1A1
SCHEMBL11446022 0.86 PKM (0.66) PKMKDM4EHSD17B10P2RX4ALDH1A1
SCHEMBL8065979 0.85 TTR (0.48) PKMKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL21962198 0.83 PKM (0.74) PKMALDH1A1HPGDCA2CA1
SCHEMBL15524940 0.82 CA12 (0.54) PKMP2RX4F10CA2CA1
SCHEMBL21814405 0.81 CA2 (0.55) PKMKDM4EHSD17B10P2RX4ALDH1A1
SCHEMBL2684958 0.80 USP2 (0.76) PKMKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL31748192 0.80 HPGD (0.54) PKMKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL8068832 0.80 PKM (0.43) PKMALDH1A1HPGDUSP2F10
SCHEMBL9196597 0.80 P2RX4 (0.47) PKMKDM4EHSD17B10P2RX4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292755-A USPA benzolyguanidines HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-08 US disclosed
US-5091394-A BENZOYLGUANIDINES, A PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-25 US disclosed