SCHEMBL9437878

SCHEMBL9437878

CCCN(CCc1ccc2c(c1)NC(=O)CO2)CCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.51
RAF1 P04049 2/20 0.47
BRAF P15056 2/20 0.47
DRD2 P14416 5/20 0.44
DRD4 P21917 3/20 0.44
DRD3 P35462 3/20 0.44
NR3C2 P08235 2/20 0.43
HTR1A P08908 5/20 0.43
HTR1D P28221 4/20 0.43
HTR1B P28222 4/20 0.43
SLC6A4 P31645 4/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAOB P27338 1/20 0.42
MAPK1 P28482 1/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437826 0.94 PARP1 (0.49) PARP1RAF1BRAFDRD2DRD4
SCHEMBL9437877 0.94 PARP1 (0.48) PARP1RAF1BRAFDRD2DRD4
SCHEMBL9437740 0.81 PARP1 (0.60) PARP1DRD2DRD4DRD3NR3C2
SCHEMBL9437919 0.80 HTR1A (0.46) DRD3HTR1AHTR1DHTR1BSLC6A4
SCHEMBL9437860 0.79 PARP1 (0.56) PARP1RAF1BRAFDRD2DRD4
SCHEMBL9437847 0.77 PARP1 (0.54) PARP1RAF1BRAFDRD2DRD4
SCHEMBL9437866 0.77 PARP1 (0.53) PARP1DRD2DRD4DRD3NR3C2
SCHEMBL12844300 0.75 PARP1 (0.78) PARP1DRD2DRD4DRD3NR3C2
SCHEMBL31033201 0.75 PARP1 (0.78) PARP1DRD2DRD4DRD3NR3C2
SCHEMBL9437886 0.75 PARP1 (0.44) PARP1DRD2DRD4DRD3NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed