SCHEMBL9437740

SCHEMBL9437740

CCCN(CCN)CCc1ccc2c(c1)NC(=O)CO2

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.60
NR3C2 P08235 3/20 0.52
MMP12 P39900 1/20 0.47
PRNP P04156 1/20 0.44
DRD4 P21917 6/20 0.43
DRD2 P14416 5/20 0.43
DRD3 P35462 3/20 0.43
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
SLC6A4 P31645 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437878 0.81 PARP1 (0.51) PARP1NR3C2DRD4DRD2DRD3
SCHEMBL9437898 0.81 PARP1 (0.68) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL12844300 0.81 PARP1 (0.78) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL31033201 0.81 PARP1 (0.78) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL9437826 0.80 PARP1 (0.49) PARP1NR3C2DRD4DRD2DRD3
SCHEMBL9437877 0.79 PARP1 (0.48) PARP1NR3C2DRD4DRD2DRD3
SCHEMBL21207261 0.79 PARP1 (0.74) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL9437820 0.79 PKM (0.54) PARP1MMP12PRNPDRD4DRD2
SCHEMBL11002313 0.78 PARP1 (0.77) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL9437774 0.77 PKM (0.52) PARP1MMP12PRNPDRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed