SCHEMBL9437882

SCHEMBL9437882

CN1C(=O)COc2cc(CCNCCCCN3C(=O)C4CCCC4C3=O)ccc21

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.44
HTR2C P28335 3/20 0.42
GABRA5 P31644 2/20 0.39
GABRA1 P14867 1/20 0.39
NMT1 P30419 3/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
SLC6A4 P31645 1/20 0.39
KCNH2 Q12809 1/20 0.39
CYP11B2 P19099 2/20 0.36
CYP11B1 P15538 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9437773 0.96 HTR1A (0.48) HTR1AHTR2CGABRA5GABRA1NMT1
SCHEMBL9437911 0.84 HTR1A (0.49) HTR1AHTR2CGABRA5GABRA1
SCHEMBL9437950 0.82 HTR1A (0.45) HTR1AHTR2CGABRA5GABRA1NMT1
SCHEMBL9437849 0.81 HTR1A (0.48) HTR1AHTR2CGABRA5GABRA1HTR1D
SCHEMBL9437784 0.80 HTR1A (0.54) HTR1AHTR2CGABRA5GABRA1
SCHEMBL9452085 0.80 HTR1A (0.47) HTR1AHTR2CGABRA5GABRA1NMT1
SCHEMBL9437710 0.80 HTR1A (0.42) HTR1AHTR2CGABRA5GABRA1NMT1
SCHEMBL9437689 0.79 HTR1A (0.50) HTR1AHTR2CGABRA5GABRA1NMT1
SCHEMBL9437900 0.79 PARP1 (0.46) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL9437879 0.78 HTR1A (0.52) HTR1AHTR2CGABRA5GABRA1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US claimed
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed