SCHEMBL9439664

SCHEMBL9439664

CCOC(=O)CC[C@@H](NC(=O)c1ccc(CCCc2c[nH]c3nc(N)nc(O)c23)s1)C(=O)OCC

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 11/20 0.56
SLC46A1 Q96NT5 9/20 0.56
SLC19A1 P41440 5/20 0.56
GART P22102 6/20 0.54
DHFR P00374 3/20 0.43
TYMS P04818 2/20 0.43
FOLR2 P14207 4/20 0.40
ATIC P31939 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9439656 1.00 FOLR1 (0.56) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439960 0.93 FOLR1 (0.57) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439954 0.93 FOLR1 (0.57) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564229 0.91 FOLR1 (0.46) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL8982495 0.86 FOLR1 (0.53) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL8982600 0.86 FOLR1 (0.53) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL8982494 0.86 FOLR1 (0.53) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9039220 0.85 DHFR (0.57) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9039215 0.85 DHFR (0.57) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439673 0.84 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed