SCHEMBL9447797

SCHEMBL9447797

O=c1cncc2ccccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP2A6 P11509 1/20 0.41
PDPK1 O15530 1/20 0.41
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
BTK Q06187 1/20 0.38
NQO2 P16083 1/20 0.37
EGFR P00533 1/20 0.37
GSTP1 P09211 1/20 0.35
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
CYP17A1 P05093 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4452628 0.69 CYP2A6 (0.47) CYP1A2CYP2A6GRIN2DGRIN3BGRIN1
Anthracene SCHEMBL29011110 0.68 CYP19A1 (0.50) CYP1A2CYP2A6PDPK1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL5243070 0.67 CYP2A6 (0.44) CYP1A2CYP2A6GRIN2DGRIN3BGRIN1
SCHEMBL7905240 0.66 GSTP1 (0.48) CYP1A2CYP2A6GRIN2DGRIN3BGRIN1
SCHEMBL445029 0.65 CLK1 (0.52) CYP1A2CYP11B1CYP11B2CYP17A1CYP19A1
SCHEMBL7427641 0.64 CYP1A2 (0.48) CYP1A2CYP2A6PDPK1BTKEGFR
Naphthalene SCHEMBL7327012 0.64 TNF (0.48) CYP1A2CYP2A6EGFRCYP11B1CYP11B2
Isoquinoline SCHEMBL1536317 0.64 TNF (0.48) CYP1A2CYP2A6EGFRCYP11B1CYP11B2
Isoquinoline SCHEMBL29355164 0.64 TNF (0.48) CYP1A2CYP2A6EGFRCYP11B1CYP11B2
Isoquinoline SCHEMBL9654 0.64 TNF (0.48) CYP1A2CYP2A6EGFRCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210082-A 2-BENZAZEPINES WITH 5- AND 6-MEMBERED HETEROCYCLIC RINGS TO TREAT PAIN AND ANXIETY DISORDERS MERCK & CO., INC. (US) 1993-05-11 US disclosed