SCHEMBL9448372

SCHEMBL9448372

COCCOc1cc(C(N)=O)ccc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.51
TSHR P16473 2/20 0.45
CHEK2 O96017 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 4/20 0.42
HTT P42858 1/20 0.42
CHEK1 O14757 1/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 2/20 0.41
NNMT P40261 1/20 0.41
PARP10 Q53GL7 1/20 0.41
RAB9A P51151 1/20 0.41
IKBKB O14920 1/20 0.41
OPRK1 P41145 1/20 0.41
PRSS1 P07477 1/20 0.41
SMPD1 P17405 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23792950 0.86 TSHR (0.50) TSHRALDH1A1HPGDKMT2AHTT
SCHEMBL6941556 0.84 MAPK1 (0.72) MAPK1TSHRHPGDTP53PRSS1
SCHEMBL17129602 0.84 L3MBTL1 (0.57) TSHRTDP1L3MBTL1KDM4EALDH1A1
SCHEMBL15101072 0.82 MAPK1 (0.69) MAPK1TSHRKDM4EKMT2AHTT
SCHEMBL30151541 0.80 MAPK1 (0.50) MAPK1CHEK2KDM4EALDH1A1HPGD
SCHEMBL3340955 0.80 MAPK1 (0.60) MAPK1TSHRL3MBTL1ALDH1A1KMT2A
SCHEMBL8901308 0.79 MAPK1 (0.49) MAPK1CHEK2KDM4EALDH1A1HPGD
SCHEMBL31053926 0.78 MAPK1 (0.63) MAPK1TSHRKMT2ATP53MEN1
SCHEMBL2936694 0.78 TSHR (0.53) TSHRTDP1ALDH1A1HPGDKMT2A
SCHEMBL2934574 0.77 TDP1 (0.52) TSHRTDP1L3MBTL1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5215738-A Used for destroying hypoxic tumor cells SRI INTERNATIONAL (US) 1993-06-01 US disclosed
WO-1986006628-A1 BENZAMIDE AND NICOTINAMIDE RADIOSENSITIZERS SRI INTERNATIONAL (US) 1986-11-20 WO disclosed