SCHEMBL9448545

SCHEMBL9448545

CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](CC(=O)O)NC(=O)CNC(=O)[C@@H](N)CCCNC(=N)N

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 3/20 0.42
KEAP1 Q14145 1/20 0.41
NPY4R P50391 8/20 0.40
NPY1R P25929 5/20 0.40
NPY2R P49146 4/20 0.40
NPY5R Q15761 4/20 0.40
OPRL1 P41146 2/20 0.40
TFPI P10646 1/20 0.39
CXCR4 P61073 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30974097 0.89 GLO1 (0.41) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL14028314 0.88 NOD1 (0.41) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL31349358 0.88 NPY4R (0.40) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL31031613 0.88 NOD1 (0.43) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL17955408 0.88 NPY4R (0.44) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL13496859 0.87 NPY4R (0.40) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL7394659 0.87 NPY4R (0.40) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL17732657 0.84 NPY4R (0.40) BMP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL29642947 0.84 TFPI (0.44) KEAP1NPY4RNPY1RNPY2RNPY5R
SCHEMBL30521941 0.83 OPRL1 (0.43) NPY4RNPY1RNPY2RNPY5ROPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522081-A4 INHIBITION OF DISEASE ASSOCIATED WITH IMMUNODEFICIENCY VIRUS INFECTION 1993-06-16 EP disclosed
EP-0522081-A1 INHIBITION OF DISEASE ASSOCIATED WITH IMMUNODEFICIENCY VIRUS INFECTION SMITHKLINE BEECHAM CORPORATION (US) 1993-01-13 EP disclosed
WO-1991015224-A1 INHIBITION OF DISEASE ASSOCIATED WITH IMMUNODEFICIENCY VIRUS INFECTION SMITHKLINE BEECHAM CORPORATION (US) 1991-10-17 WO disclosed