SCHEMBL9449028

SCHEMBL9449028

OCc1ccc2c(C3CN4CCC3CC4)c[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.52
NOS1 P29475 3/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C19 P33261 1/20 0.52
NOS2 P35228 1/20 0.52
IDO1 P14902 1/20 0.39
SLC6A4 P31645 2/20 0.38
CHRNA7 P36544 2/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
APP P05067 1/20 0.36
DRD2 P14416 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ATM Q13315 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9448835 0.90 NOS3 (0.55) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448897 0.83 NOS3 (0.54) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448970 0.81 NOS3 (0.52) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL4311896 0.78 HTR2C (0.55) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448872 0.78 NOS3 (0.49) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9449311 0.76 IMPDH2 (0.50) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448887 0.75 NOS3 (0.48) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL3546179 0.75 CYP3A4 (0.56) NOS3NOS1CYP3A4CYP2C19NOS2
SCHEMBL9448885 0.75 NOS3 (0.46) NOS3NOS1CYP3A4CYP2C19NOS2
Hydrochloric Acid SCHEMBL9449059 0.74 CYP3A4 (0.55) NOS3NOS1CYP3A4CYP2C19NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5227386-A INDOLE DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-07-13 US disclosed