SCHEMBL9449952

SCHEMBL9449952

CN(C(=O)Cc1ccc(OCc2ccccc2)cc1)C(CN1CCC(O)C1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 16/20 0.71
OPRM1 P35372 13/20 0.71
OPRD1 P41143 13/20 0.71
CYP2D6 P10635 9/20 0.71
CCR5 P51681 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17776365 0.90 OPRK1 (0.77) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL17776358 0.90 OPRK1 (0.77) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL7945544 0.90 OPRK1 (0.77) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL9450205 0.90 OPRK1 (0.73) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL9450203 0.88 OPRK1 (0.75) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL8720262 0.87 OPRK1 (0.78) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL9450279 0.86 OPRK1 (0.79) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL17776366 0.86 OPRK1 (0.76) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL17776369 0.86 OPRK1 (0.79) OPRK1OPRM1OPRD1CYP2D6
SCHEMBL17776372 0.86 OPRK1 (0.79) OPRK1OPRM1OPRD1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5232978-A 1-(2-arylethyl)-pyrrolidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-08-03 US disclosed
EP-0483580-A2 1-(2-Arylethyl)-pyrrolidine MERCK PATENT GmbH (DE) 1992-05-06 EP disclosed