SCHEMBL9450845

SCHEMBL9450845

FC(F)(F)c1ccc([C@H]2CC[C@H](CCC3CCC([C@H]4CC[C@H](/C=C/Cl)CC4)CC3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.47
ESR2 Q92731 5/20 0.36
IDO1 P14902 1/20 0.35
CYP2C9 P11712 3/20 0.35
ESR1 P03372 3/20 0.35
CYP3A4 P08684 2/20 0.35
CHRM2 P08172 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CNR1 P21554 1/20 0.35
MAOB P27338 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
DGAT1 O75907 2/20 0.33
SOAT1 P35610 1/20 0.33
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962970 0.96 HTR2C (0.50) HTR2CESR2IDO1CYP2C9ESR1
SCHEMBL8962978 0.96 HTR2C (0.50) HTR2CESR2IDO1CYP2C9ESR1
SCHEMBL8962960 0.93 HTR2C (0.53) HTR2CCNR1MAOB
SCHEMBL8963017 0.89 HTR2C (0.57) HTR2CCNR1MAOB
SCHEMBL8963025 0.89 HTR2C (0.57) HTR2CCNR1MAOB
SCHEMBL8962904 0.85 HTR2C (0.53) HTR2CCHRM2CHRM5MAOBDGAT1
SCHEMBL8962900 0.85 HTR2C (0.53) HTR2CCHRM2CHRM5MAOBDGAT1
SCHEMBL8968584 0.82 CYP2C9 (0.49) ESR2CYP2C9ESR1CYP3A4MAOB
SCHEMBL8963241 0.82 ESR2 (0.41) ESR2CYP2C9ESR1CYP3A4ALDH1A1
SCHEMBL9300385 0.82 ESR2 (0.41) ESR2CYP2C9ESR1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed