SCHEMBL945299

SCHEMBL945299

CSc1nc(-c2ccc(F)cc2)c(CO)c(C(C)C)n1

nearest known ligand 0.57

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GCGR P47871 19/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL944388 0.87 GCGR (0.43) GCGR
SCHEMBL14400742 0.82 GCGR (0.47) GCGR
SCHEMBL7920817 0.82 GCGR (0.46) GCGR
SCHEMBL10129581 0.80 DHODH (0.44) GCGR
SCHEMBL4449474 0.79 GCGR (0.63) GCGR
SCHEMBL12912572 0.78 RXFP1 (0.40) GCGR
SCHEMBL27984907 0.78 KMT2A (0.51)
SCHEMBL14400636 0.77 MAPT (0.37) GCGR
SCHEMBL8949822 0.77 GCGR (0.88) GCGR
SCHEMBL16429685 0.77 GCGR (0.57) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872012-B2 Pyrimidinone compounds and preparation and use thereof Zhejiang Hisun Pharma Co., Ltd. (CN) 2011-01-18 US disclosed
US-7872012-B2 Pyrimidinone compounds and preparation and use thereof Zhejiang Hisun Pharma Co., Ltd. (CN) 2011-01-18 US disclosed
EP-1845092-B1 PYRIMIDINONE COMPOUNDS, THEIR PREPARATION AND USE THEREOF YAO HUI (CN) 2010-09-01 EP disclosed
US-20080280930-A1 Pyrimidinone Compounds and Preparation and Use Thereof Yao, Hui (CN) 2008-11-13 US disclosed
US-20080280930-A1 Pyrimidinone Compounds and Preparation and Use Thereof Yao, Hui (CN) 2008-11-13 US disclosed
US-7371759-B2 HMG-CoA reductase inhibitors and method BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-13 US disclosed
US-7371759-B2 HMG-CoA reductase inhibitors and method BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-13 US disclosed
EP-1845092-A1 PYRIMIDINONE COMPOUNDS, THEIR PREPARATION AND USE THEREOF Yao, Hui (CN) 2007-10-17 EP disclosed
EP-1845092-A1 PYRIMIDINONE COMPOUNDS, THEIR PREPARATION AND USE THEREOF Yao, Hui (CN) 2007-10-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280930-A1 Pyrimidinone Compounds and Preparation and Use Thereof HMGCR, PSEN1, DHPS GCGR 1827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.