SCHEMBL10129581

SCHEMBL10129581

CSc1nc(-c2ccc(F)cc2)c(C(=O)O)c(C(C)C)n1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 12/20 0.44
GCGR P47871 1/20 0.41
RXFP1 Q9HBX9 2/20 0.40
MAPT P10636 1/20 0.37
TP53 P04637 1/20 0.37
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
PPARG P37231 1/20 0.36
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945897 0.86 GCGR (0.55) DHODHGCGRRXFP1MAPTTP53
SCHEMBL3589 0.83 ALDH1A1 (0.44) GCGRMAPTTP53ALDH1A1L3MBTL1
SCHEMBL10153184 0.82 GCGR (0.43) DHODHGCGRPDE10A
SCHEMBL6082682 0.81 ADORA2A (0.44) DHODHGCGRPDE10A
SCHEMBL27519225 0.81 DHODH (0.45) DHODHRXFP1MAPTALDH1A1L3MBTL1
SCHEMBL945299 0.80 GCGR (0.57) GCGR
SCHEMBL7920817 0.79 GCGR (0.46) GCGRALDH1A1L3MBTL1CYP2C19
SCHEMBL10433875 0.79 HMGCR (0.48) DHODHGCGRMAPTTP53ALDH1A1
SCHEMBL10434011 0.79 HMGCR (0.44) DHODHGCGRALDH1A1PDE10A
SCHEMBL28300700 0.79 ADORA1 (0.47) DHODHGCGRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012013325-A1 PROCESS FOR THE PREPARATION OF KEY INTERMEDIATES FOR THE SYNTHESIS OF STATINS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF LEK PHARMACEUTICALS D.D. (SI) 2012-02-02 WO disclosed