SCHEMBL945540

SCHEMBL945540

CCOC(=O)CC1CCn2c1nc1cc(C#N)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP14 P54578 3/20 0.39
S1PR1 P21453 1/20 0.37
ITK Q08881 1/20 0.37
F2 P00734 2/20 0.37
MAPT P10636 2/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.36
GRM5 P41594 1/20 0.36
HSD11B1 P28845 1/20 0.36
CYP11B2 P19099 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014862 0.85 MIF (0.40) F2TSHRHSD17B10KDM4EALDH1A1
SCHEMBL10532632 0.68 PPARA (0.47) CYP1A2GRM5CYP11B2
SCHEMBL22070895 0.68 CYP11B1 (0.42) MAPTL3MBTL1KDM4EALDH1A1HPGD
SCHEMBL12320236 0.68 S1PR1 (0.46) S1PR1ALDH1A1GAAMAPK1
SCHEMBL933742 0.67 ALDH1A1 (0.42) USP14MAPTALDH1A1GAAMAPK1
SCHEMBL9588938 0.66 FFAR4 (0.40) S1PR1MAPTTSHRHSD17B10KDM4E
SCHEMBL7753345 0.66 USP14 (0.52) USP14MAPTL3MBTL1KDM4EALDH1A1
SCHEMBL950210 0.65 S1PR1 (0.58) S1PR1
SCHEMBL2018070 0.65 GAA (0.37) S1PR1MAPTTSHRHSD17B10KDM4E
SCHEMBL2470686 0.64 MAPT (0.48) MAPTTSHRHSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005290-A1 DISUBSTITUTED OXADIAZOLE DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed