SCHEMBL9458013

SCHEMBL9458013

COc1cccc2c1[C@H]1CCNC[C@@H]1C2

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 11/20 0.44
GNAI3 P08754 1/20 0.42
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9035226 1.00 HTR1A (0.44) HTR1AGNAI3HTR2CHTR2BHTR2A
SCHEMBL9458029 1.00 HTR1A (0.44) HTR1AGNAI3HTR2CHTR2BHTR2A
SCHEMBL9035221 1.00 HTR1A (0.44) HTR1AGNAI3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL9035512 0.99 HTR1A (0.43) HTR1AGNAI3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL9457774 0.99 HTR1A (0.43) HTR1AGNAI3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL9035515 0.99 HTR1A (0.43) HTR1AGNAI3HTR2CHTR2BHTR2A
Hydrochloric Acid SCHEMBL9035522 0.99 HTR1A (0.43) HTR1AGNAI3HTR2CHTR2BHTR2A
SCHEMBL7844867 0.77 HTR2C (0.38) HTR1AGNAI3HTR2C
SCHEMBL7844871 0.77 HTR2C (0.38) HTR1AGNAI3HTR2C
SCHEMBL8139163 0.75 HTR1A (0.49) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422134-A1 5-HT SELECTIVE AGENTS. ABBOTT LAB (US) 1991-04-17 EP claimed
WO-1990006927-A1 5-HT SELECTIVE AGENTS ABBOTT LABORATORIES (US) 1990-06-28 WO claimed
US-5244888-A Hexahydroindenopyrroles and hexahydrobenzisoindoles ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
US-5049564-A Hypotensive, 5-hydroxytryptamine ABBOTT LABORATORIES (US) 1991-09-17 US disclosed
EP-0422134-A1 5-HT SELECTIVE AGENTS. ABBOTT LAB (US) 1991-04-17 EP disclosed
WO-1990006927-A1 5-HT SELECTIVE AGENTS ABBOTT LABORATORIES (US) 1990-06-28 WO disclosed