SCHEMBL9458430

SCHEMBL9458430

CC(C)(C)c1cccc(Oc2cc(F)cc(C3(O)CCOCC3)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 8/20 0.43
MMP13 P45452 2/20 0.38
MMP2 P08253 1/20 0.38
MMP3 P08254 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP14 P50281 1/20 0.38
CTSD P07339 1/20 0.37
BACE1 P56817 1/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
MMP1 P03956 1/20 0.37
P2RY1 P47900 1/20 0.36
S1PR2 O95136 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458371 0.87 ALOX5 (0.45) ALOX5MMP13MMP2MMP3MMP9
SCHEMBL9458568 0.79 ALOX5 (0.48) ALOX5MMP13MMP1
SCHEMBL9458556 0.75 ALOX5 (0.37) ALOX5S1PR2
SCHEMBL18210658 0.72 CYP3A4 (0.50) MMP2MMP3MMP9MMP14SLC6A2
SCHEMBL9458313 0.71 OPRL1 (0.43) ALOX5MMP13MMP2MMP3MMP9
SCHEMBL31070675 0.71 EPAS1 (0.46) P2RY1CYP3A4CYP2C9CYP2C19
SCHEMBL7479848 0.71 HDAC3 (0.43) ALOX5SLC6A2SLC6A3
SCHEMBL9458222 0.71 ALOX5 (0.36) ALOX5MMP13CTSDBACE1MMP1
SCHEMBL8551875 0.70 ALOX5 (0.59) ALOX5PTGS1PTGS2
SCHEMBL18118971 0.69 CYP3A4 (0.59) CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed