SCHEMBL9458496

SCHEMBL9458496

FC(F)(F)c1cc(Br)cc(Sc2ccc(CBr)cc2)c1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
NOTUM Q6P988 1/20 0.33
CNR1 P21554 1/20 0.32
PARK7 Q99497 1/20 0.32
ACP1 P24666 1/20 0.31
TAS2R14 Q9NYV8 1/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458299 0.82 MAOB (0.35) S1PR1S1PR3NOTUMCNR1SLC6A2
SCHEMBL9458506 0.81 MLYCD (0.47) S1PR1S1PR3NOTUM
SCHEMBL15207303 0.78 MAOB (0.42)
SCHEMBL9853038 0.76 NOTUM (0.34) NOTUMTAS2R14
SCHEMBL9458604 0.75 CYP2A6 (0.40) S1PR1S1PR3NOTUMTAS2R14SLC6A2
SCHEMBL9853033 0.74 SLC6A4 (0.38) PARK7SLC6A2SLC6A4SLC6A3
SCHEMBL3591051 0.74 IDO1 (0.41) S1PR1S1PR3NOTUMCNR1PARK7
SCHEMBL29738521 0.74 IDO1 (0.41) S1PR1S1PR3NOTUMCNR1PARK7
SCHEMBL9457966 0.74 CYP19A1 (0.37) S1PR1S1PR3NOTUMSLC6A2SLC6A4
SCHEMBL7561792 0.73 TSHR (0.48) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed