SCHEMBL9458299

SCHEMBL9458299

N#CCc1ccc(Sc2cc(Br)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.35
MAOA P21397 2/20 0.35
PTPRC P08575 1/20 0.33
PTPN1 P18031 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
RXRA P19793 2/20 0.32
RXRG P48443 2/20 0.32
RXRB P28702 1/20 0.32
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
AR P10275 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
MCL1 Q07820 1/20 0.30
CNR1 P21554 1/20 0.30
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458496 0.82 S1PR1 (0.33) S1PR1S1PR3SLC6A2SLC6A4SLC6A3
SCHEMBL9457966 0.78 CYP19A1 (0.37) MAOBMAOAMEN1ALDH1A1KMT2A
SCHEMBL21854601 0.77 NOTUM (0.37) PTPRCPTPN1RXRARXRGRXRB
SCHEMBL9458506 0.76 MLYCD (0.47) MEN1ALDH1A1KMT2AS1PR1S1PR3
SCHEMBL15207303 0.73 MAOB (0.42) MAOBMAOAMCL1
SCHEMBL9458055 0.73 WDR5 (0.34) MAOBMAOAMEN1ALDH1A1KMT2A
SCHEMBL246959 0.71 TAAR1 (0.48) MAOBALDH1A1KMT2A
SCHEMBL9458604 0.71 CYP2A6 (0.40) PTPN1MEN1ALDH1A1KMT2AS1PR1
SCHEMBL7594667 0.69 RXRA (0.54) MAOBRXRARXRGRXRB
SCHEMBL9168708 0.68 MAOA (0.55) MAOBMAOAALDH1A1KMT2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed