SCHEMBL9458759

SCHEMBL9458759

Nc1c(C=O)cnn1-c1ccc(OC(F)(F)F)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 2/20 0.37
MCHR1 Q99705 2/20 0.37
MAPK1 P28482 2/20 0.36
MAPT P10636 2/20 0.36
RECQL P46063 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CHRM5 P08912 6/20 0.35
SCN9A Q15858 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
GMNN O75496 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458706 0.79 KMT2A (0.44) NPBWR1MCHR1MAPK1MAPTRECQL
SCHEMBL1884450 0.74 FGFR1 (0.45) SCN9ANPC1RAB9ALMNAGAA
SCHEMBL3148079 0.73 TDP1 (0.50) MAPK1CHRM5SCN9ANPC1RAB9A
SCHEMBL6201722 0.70 FFAR4 (0.41) MAPK1CHRM5SCN9ANPC1RAB9A
SCHEMBL21339745 0.70 NPC1 (0.47) MAPK1SCN9ANPC1RAB9AGMNN
SCHEMBL10737936 0.69 CHRM5 (0.35) NPBWR1MCHR1MAPK1MAPTRECQL
SCHEMBL10738468 0.69 TRPA1 (0.34) NPBWR1MCHR1MAPK1MAPTRECQL
SCHEMBL14843789 0.69 HCRTR1 (0.40) CHRM5SCN5AHCRTR1
SCHEMBL28304122 0.69 SMURF1 (0.41) NPBWR1MCHR1MAPK1MAPTRECQL
SCHEMBL15332944 0.68 TDP1 (0.49) L3MBTL1LMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256634-A Herbicidal agents based on pyrazole derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-10-26 US disclosed
US-5104439-A HERBICIDAL AGENTS BASED ON PYRAZOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-14 US disclosed
EP-0154115-B1 HERBICIDAL COMPOSITIONS BASED ON DERIVATIVES OF PYRAZOLES BAYER AG (DE) 1988-10-26 EP disclosed
US-4614533-A Herbicidal 5-amino-1-phenylpyrazoles BAYER AKTIENGESELLSCHAFT (DE) 1986-09-30 US disclosed
EP-0154115-A1 Herbicidal compositions based on derivatives of pyrazoles BAYER AG (DE) 1985-09-11 EP disclosed