SCHEMBL9460875

SCHEMBL9460875

C=Cc1ccc(OCCC[Si](C)(OCC)OCC)cc1.C=Cc1cccc(OCCC[Si](C)(OC)OC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.40
CHRNB2 P17787 3/20 0.40
CHRNB4 P30926 3/20 0.40
CHRNA3 P32297 3/20 0.40
CHRNA4 P43681 3/20 0.40
TLR4 O00206 1/20 0.38
TLR2 O60603 1/20 0.38
AHR P35869 1/20 0.36
NPC1 O15118 4/20 0.35
POLB P06746 4/20 0.35
RAB9A P51151 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 3/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
MAPK1 P28482 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9315267 0.91 TLR4 (0.41) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL8776506 0.88 TLR4 (0.40) CHRNA7TLR4TLR2NPC1POLB
SCHEMBL1269637 0.86 CHRNA7 (0.51) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL4372162 0.83 CHRNA7 (0.50) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9316433 0.81 TLR4 (0.41) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9316455 0.80 TLR4 (0.42) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL15505269 0.79 CHRNA7 (0.53) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9315501 0.78 TLR4 (0.40) CHRNA7TLR4TLR2NPC1POLB
SCHEMBL9461719 0.78 CHRNA7 (0.46) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9315977 0.77 NPC1 (0.43) CHRNA7TLR4TLR2NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210252-A 3-(VINYLPHENYLOXY)PROPYLSILANE COMPOUND SHIN-ETSU CHEMICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5196591-A PROCESS FOR THE PRODUCTION OF POLYNUCLEAR AROMATIC POLYAMINES BAYER AKTIENGESELLSCHAFT (DE) 1993-03-23 US disclosed