Bromide

Bromide

SCHEMBL9464396

Br.NCC(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A known ✓ P08908 2/20 0.41
DPP4 P27487 9/20 0.54
PREP P48147 1/20 0.54
FAP Q12884 1/20 0.54
DPP8 Q6V1X1 1/20 0.54
DPP9 Q86TI2 1/20 0.54
ACE P12821 2/20 0.44
HTR7 P34969 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9464510 1.00 DPP4 (0.54) DPP4PREPFAPDPP8DPP9
SCHEMBL8772871 0.98 DPP4 (0.56) DPP4PREPFAPDPP8DPP9
SCHEMBL8772866 0.98 DPP4 (0.56) DPP4PREPFAPDPP8DPP9
Hydrochloric Acid SCHEMBL19692659 0.96 DPP4 (0.54) DPP4PREPFAPDPP8DPP9
Hydrochloric Acid SCHEMBL29548868 0.96 DPP4 (0.54) DPP4PREPFAPDPP8DPP9
SCHEMBL10884099 0.84 DPP4 (0.54) DPP4ACEHTR1AHTR7
Glycyl Proline SCHEMBL155067 0.83 ACE (0.62) DPP4PREPFAPDPP8DPP9
Glycyl Proline SCHEMBL30051559 0.83 ACE (0.62) DPP4PREPFAPDPP8DPP9
SCHEMBL1493753 0.83 DPP4 (0.47) DPP4ACEHTR1AHTR7
Glycyl Proline SCHEMBL155066 0.83 ACE (0.62) DPP4PREPFAPDPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294668-B1 (2-CYANO-2-OXIMINOACETYL)-AMINO ACID DERIVATIVES BAYER AG (DE) 1993-04-07 EP disclosed
EP-0294667-B1 (2-CYANO-2-OXIMINOACETYL)-AMINO ACID DERIVATIVES BAYER AG (DE) 1993-03-17 EP disclosed
US-5189061-A Fungicide BAYER AKTIENGESELLSCHAFT (DE) 1993-02-23 US disclosed
US-5026710-A Fungicides BAYER AKTIENGESELLSCHAFT (DE) 1991-06-25 US disclosed
US-4963548-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1990-10-16 US disclosed
EP-0294668-A2 (2-cyano-2-oximinoacetyl)-amino acid derivatives BAYER AG (DE) 1988-12-14 EP disclosed
EP-0294667-A2 (2-cyano-2-oximinoacetyl)-amino acid derivatives BAYER AG (DE) 1988-12-14 EP disclosed