SCHEMBL9466832

SCHEMBL9466832

C1=C(c2ccccc2)CCN(CCCCc2ccncc2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 1.00
DRD2 P14416 1/20 0.59
DRD4 P21917 1/20 0.59
DRD3 P35462 1/20 0.59
PARP1 P09874 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9719779 0.99 SIGMAR1 (0.97) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL9473840 0.96 SIGMAR1 (0.92) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL9467083 0.86 SIGMAR1 (0.76) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL9466872 0.85 SIGMAR1 (1.00) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL10974243 0.84 SIGMAR1 (0.72) SIGMAR1DRD2DRD4DRD3PARP1
Hydrochloric Acid SCHEMBL10937128 0.83 SIGMAR1 (0.71) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL9466973 0.83 SIGMAR1 (1.00) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL9377531 0.82 SIGMAR1 (1.00) SIGMAR1PARP1
SCHEMBL9467457 0.81 SIGMAR1 (0.68) SIGMAR1DRD2DRD4DRD3PARP1
SCHEMBL10970684 0.81 SIGMAR1 (0.67) SIGMAR1DRD2DRD4DRD3PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed