SCHEMBL9466872

SCHEMBL9466872

C1=C(c2ccccn2)CCN(CCCCc2ccncc2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 1.00
TMEM97 Q5BJF2 1/20 0.50
DRD4 P21917 2/20 0.48
PPARG P37231 1/20 0.45
PPARA Q07869 1/20 0.45
PARP1 P09874 1/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9467081 0.87 SIGMAR1 (0.78) SIGMAR1TMEM97DRD4DRD2DRD3
SCHEMBL9466832 0.85 SIGMAR1 (1.00) SIGMAR1DRD4PARP1DRD2DRD3
SCHEMBL9719779 0.84 SIGMAR1 (0.97) SIGMAR1DRD4PARP1DRD2DRD3
SCHEMBL9467634 0.82 SIGMAR1 (0.69) SIGMAR1TMEM97DRD4PPARGPPARA
SCHEMBL9473840 0.81 SIGMAR1 (0.92) SIGMAR1TMEM97DRD4PARP1DRD2
SCHEMBL9466973 0.79 SIGMAR1 (1.00) SIGMAR1TMEM97DRD4PPARGPPARA
SCHEMBL9467235 0.76 SIGMAR1 (1.00) SIGMAR1TMEM97DRD2
SCHEMBL6969008 0.76 DRD4 (0.61) SIGMAR1DRD4PPARGPPARADRD2
SCHEMBL25124555 0.75 SIGMAR1 (0.60) SIGMAR1DRD4PPARGPPARADRD2
SCHEMBL10974243 0.73 SIGMAR1 (0.72) SIGMAR1DRD4PPARGPPARAPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US claimed
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed