SCHEMBL9468366

SCHEMBL9468366

CC1=C(c2ccc(Cl)cc2)n2ncc(C#N)c2N(C(=O)CCl)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 4/20 0.34
GAA P10253 3/20 0.34
LMNA P02545 2/20 0.34
HPGD P15428 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
HSD17B3 P37058 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
POLB P06746 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9468410 0.88 RXRA (0.47) RXRARXRBRXRGALDH1A1KDM4E
SCHEMBL10694331 0.83 DRD4 (0.44) ALDH1A1KMT2AMEN1
SCHEMBL9468461 0.81 KDM4E (0.40) RXRARXRBRXRGCYP1A2CYP3A4
SCHEMBL9468042 0.81 DRD4 (0.43) RXRARXRBRXRGALDH1A1KDM4E
SCHEMBL9468824 0.79 RXRA (0.35) RXRARXRBRXRGCYP1A2CYP3A4
SCHEMBL9468364 0.77 DRD4 (0.40) ALDH1A1KDM4ENPC1RAB9AL3MBTL1
SCHEMBL9468091 0.74 RXRA (0.41) RXRARXRBRXRGALDH1A1LMNA
SCHEMBL9468869 0.71 KMT2A (0.43) RXRARXRBRXRGALDH1A1KDM4E
SCHEMBL9468331 0.70 KDM4E (0.39) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL9468714 0.69 UBE2M (0.38) RXRARXRBRXRGALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5219857-A Method of treating cognitive and related neural behavioral problems AMERICAN CYANAMID COMPANY (US) 1993-06-15 US disclosed
US-5126340-A Antidepressants AMERICAN CYANAMID COMPANY (US) 1992-06-30 US disclosed
US-4963553-A TREATING COGNITIVE AND NEURAL BEHAVIORAL PROBLEMS IN MAMMALS AMERICAN CYANAMID CO. (US) 1990-10-16 US disclosed
EP-0264773-A1 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1988-04-27 EP disclosed