SCHEMBL9475779

SCHEMBL9475779

CC1=C(C(=O)O)C(c2ccccc2[N+](=O)[O-])N(C(=O)C2CCCC2)C(=S)N1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1D Q01668 8/20 0.58
CACNA1F O60840 7/20 0.58
CACNA1S Q13698 7/20 0.58
CACNA1C Q13936 7/20 0.58
MAPT P10636 4/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 3/20 0.43
CACNA1B Q00975 2/20 0.43
POLB P06746 2/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ABCC4 O15439 1/20 0.43
PLIN1 O60240 1/20 0.43
GMNN O75496 1/20 0.43
KCNK2 O95069 1/20 0.43
ABCB11 O95342 1/20 0.43
GSR P00390 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476298 0.90 CACNA1D (0.48) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL9475008 0.86 CACNA1F (0.66) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL9475596 0.78 CACNA1C (0.68) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL9475454 0.77 CACNA1D (0.53) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL10557782 0.77 CACNA1F (0.54) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL10358732 0.76 CACNA1D (0.58) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL9477065 0.75 CACNA1F (0.67) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL4608748 0.70 CACNA1C (0.73) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL612520 0.70 CACNA1C (0.73) CACNA1DCACNA1FCACNA1SCACNA1CMAPT
SCHEMBL9474962 0.70 CACNA1F (0.63) CACNA1DCACNA1FCACNA1SCACNA1CMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202330-A Hypotensive and cardiovascular agent, reduces blood pressure in mammals E. R. SQUIBB & SONS, INC. (US) 1993-04-13 US disclosed
EP-0204317-A2 2-Thio or oxo-4-aryl or heterocyclo-1,5(2H)-pyrimidinedicarboxylic acid diesters and 3-acyl-5-pyrimidinecarboxylic acids and esters E.R. Squibb & Sons, Inc. (US) 1986-12-10 EP disclosed