SCHEMBL9479079

SCHEMBL9479079

N#C/C=C/c1ccc(CBr)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
FDPS P14324 1/20 0.40
ENPP2 Q13822 1/20 0.37
AKR1C3 P42330 2/20 0.36
TRPA1 O75762 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
ESR1 P03372 1/20 0.36
CYP1A1 P04798 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP1B1 Q16678 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9479084 1.00 KDM4E (0.50) KDM4EFDPSENPP2AKR1C3TRPA1
SCHEMBL10846493 0.79 KDM4E (0.64) KDM4EFDPSENPP2ALDH1A1ESR1
SCHEMBL9004477 0.79 TRPA1 (0.48) KDM4ETRPA1ALDH1A1TSHRCES2
SCHEMBL9004476 0.79 TRPA1 (0.48) KDM4ETRPA1ALDH1A1TSHRCES2
SCHEMBL3144474 0.79 KDM4E (0.64) KDM4EFDPSENPP2ALDH1A1ESR1
SCHEMBL10506198 0.79 KDM4E (0.50) KDM4EFDPSENPP2AKR1C3ESR1
SCHEMBL11444224 0.79 KDM4E (0.55) KDM4EFDPSENPP2AKR1C3ALDH1A1
SCHEMBL21457286 0.79 KDM4E (0.55) KDM4EFDPSENPP2AKR1C3ALDH1A1
SCHEMBL18160984 0.79 KDM4E (0.50) KDM4EFDPSENPP2AKR1C3ESR1
SCHEMBL10506200 0.79 KDM4E (0.50) KDM4EFDPSENPP2AKR1C3ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5234942-A Treating allergic pulmonary disorders, asthma ICI AMERICAS INC. (US) 1993-08-10 US disclosed
US-4997844-A Compounds for the treatment of allergic or inflammatory diseases or shock conditions ICI AMERICAS INC. (US) 1991-03-05 US disclosed
EP-0179619-B1 HETEROCYCLIC AMIDES ICI AMERICAS INC. (US) 1990-09-05 EP disclosed
US-4847404-A FLUORESCENT DYES, OPTICAL BRIGHTENERS CIBA-GEIGY CORPORATION (US) 1989-07-11 US disclosed
US-4780558-A CHEMICAL INTERMEDIATES FOR STILBENE FLUORESCENT WHITENING AGENTS CIBA-GEIGY CORPORATION (US) 1988-10-25 US disclosed
EP-0179619-A1 Heterocyclic amides ICI AMERICAS INC. (US) 1986-04-30 EP disclosed
US-4482496-A WHITENERS CIBA-GEIGY CORPORATION (US) 1984-11-13 US disclosed
US-4366189-A WHITENERS CIBA-GEIGY CORPORATION (US) 1982-12-28 US disclosed
US-4226878-A ANTIINFLAMMATORY, HYPOTENSIVES, ANTIHISTAMINES KISSEI PHARMACEUTICAL CO., LTD. (JP) 1980-10-07 US disclosed