SCHEMBL9482986

SCHEMBL9482986

CON=Cc1c(C(C)C)nc(C(C)C)c(C=O)c1-c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GCGR P47871 19/20 0.47
ESR1 P03372 1/20 0.40
HMGCR P04035 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
PDE4A P27815 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9482981 1.00 GCGR (0.47) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9482135 0.88 GCGR (0.44) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9482140 0.88 GCGR (0.44) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL8949603 0.87 GCGR (0.58) GCGR
SCHEMBL9483365 0.82 GCGR (0.69) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9483362 0.82 GCGR (0.69) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL8949673 0.79 GCGR (0.50) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL14097269 0.78 GCGR (0.49) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL7077308 0.78 GCGR (0.67) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9482432 0.76 HMGCR (0.56) GCGRESR1HMGCRCHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5183897-A Certain intermediate imino-substituted pyridines BAYER AKTIENGESELLSCHAFT (DE) 1993-02-02 US disclosed
US-5064841-A HMG-COA reductase-inhibiting imino-substituted pyridines BAYER AKTIENGESELLSCHAFT (DE) 1991-11-12 US disclosed
EP-0411420-A2 Imino substituted pyridine BAYER AG (DE) 1991-02-06 EP disclosed