SCHEMBL9484150

SCHEMBL9484150

CC1(C)CCC(C)(C)c2cc(C(Br)C(Br)c3ccc(C#N)cc3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.42
RXRB P28702 5/20 0.42
RARB P10826 11/20 0.40
RARG P13631 11/20 0.40
RARA P10276 8/20 0.40
CYP26A1 O43174 3/20 0.40
CYP3A4 P08684 3/20 0.40
CRABP2 P29373 1/20 0.40
CYP26B1 Q9NR63 1/20 0.39
RXRG P48443 3/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320778 0.80 RXRA (0.35) RXRARARBRARGRARACYP26A1
SCHEMBL7931062 0.80 RXRA (0.40) RXRARXRBRARBRARGRARA
SCHEMBL7929330 0.80 RARB (0.38) RXRARXRBRARBRARGRARA
SCHEMBL7929331 0.80 RARB (0.38) RXRARXRBRARBRARGRARA
SCHEMBL2223445 0.79 RARB (0.53) RXRARXRBRARBRARGRARA
SCHEMBL9483828 0.76 RARB (0.63) RXRARXRBRARBRARGRARA
SCHEMBL11240964 0.74 RXRA (0.54) RXRARXRBRARBRARGRARA
SCHEMBL10515701 0.73 RARB (0.58) RXRARXRBRARBRARGRARA
SCHEMBL10515704 0.73 RARB (0.58) RXRARXRBRARBRARGRARA
SCHEMBL3175854 0.70 RXRA (0.57) RXRARXRBRARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256694-A For skin disorders; carcinomas BASF AKTIENGESELLSCHAFT (DE) 1993-10-26 US disclosed
US-5126371-A Precancerous skin conditions, acne, psoriasis BASF AKTEINGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-4994489-A Ester derivatives of diarylacetylenes, their compositions and their use in acne treatment BASF AKTIENGESELLSCHAFT 1991-02-19 US disclosed
EP-0176034-B1 DIARYL ACETYLENES, THEIR PREPARATION AND USE BASF Aktiengesellschaft (DE) 1989-08-30 EP disclosed
US-4806558-A Diarylacetylenes and their use in treating acne BASF AKTIENGESELLSCHAFT (DE) 1989-02-21 US disclosed
EP-0176034-A2 Diaryl acetylenes, their preparation and use BASF Aktiengesellschaft (DE) 1986-04-02 EP disclosed