SCHEMBL9484161

SCHEMBL9484161

C#Cc1ccc2c(c1)C(C)(C)C(C)C2(C)C

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.33
BACE1 P56817 3/20 0.32
CTSD P07339 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9484539 0.75 RARB (0.38) BACE1BACE2
SCHEMBL6477078 0.73 CYP26A1 (0.33) BACE1CTSDBACE2
SCHEMBL9483415 0.72 RARB (0.38) RXRA
SCHEMBL1468020 0.71 RXRA (0.39) RXRA
SCHEMBL29870908 0.71 RXRA (0.39) RXRA
SCHEMBL9484220 0.71 RARB (0.41) RXRABACE1CTSDBACE2
SCHEMBL2223568 0.71 RARB (0.53) RXRA
SCHEMBL10335841 0.69 ADRA2A (0.35) RXRABACE1CTSDBACE2
SCHEMBL15309162 0.69 HDAC8 (0.32)
SCHEMBL5594371 0.69 CYP26A1 (0.31) BACE1CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256694-A For skin disorders; carcinomas BASF AKTIENGESELLSCHAFT (DE) 1993-10-26 US disclosed
US-5126371-A Precancerous skin conditions, acne, psoriasis BASF AKTEINGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-4994489-A Ester derivatives of diarylacetylenes, their compositions and their use in acne treatment BASF AKTIENGESELLSCHAFT 1991-02-19 US disclosed
US-4806558-A Diarylacetylenes and their use in treating acne BASF AKTIENGESELLSCHAFT (DE) 1989-02-21 US disclosed