SCHEMBL9488351

SCHEMBL9488351

COc1cc(C(=O)O)ccc1C(C)c1c[nH]c2ccc(CC(C)NC(=O)N(C)C)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.39
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36
TRPV1 Q8NER1 2/20 0.35
TSHR P16473 1/20 0.34
ACHE P22303 1/20 0.34
NR1H4 Q96RI1 1/20 0.33
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA7 P43166 1/20 0.33
TPMT P51580 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9488888 0.93 ACACB (0.39) ACACBROCK2ROCK1MTNR1AMTNR1B
SCHEMBL9488414 0.86 TRPV1 (0.41) MTNR1AMTNR1BTRPV1ACHEKMT2A
SCHEMBL9488311 0.84 ACACB (0.37) ACACBROCK2ROCK1TSHR
SCHEMBL9489442 0.83
SCHEMBL9489374 0.83 MGAM (0.43) ROCK2ROCK1ACHE
SCHEMBL8536466 0.82 CA12 (0.47) MTNR1AMTNR1BTRPV1TSHRCA12
SCHEMBL9373824 0.79 PRSS1 (0.38) MTNR1AMTNR1BTSHRKMT2A
SCHEMBL9373727 0.79 PPARA (0.41) MTNR1AMTNR1BTRPV1
SCHEMBL8533902 0.79 GPR84 (0.46) MTNR1AMTNR1BTRPV1TSHRKMT2A
SCHEMBL8533040 0.79 GPR84 (0.46) MTNR1AMTNR1BTRPV1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337766-B1 HETERA-ALIPHATIC CARBOXAMIDES ICI AMERICAS INC. (US) 1993-03-10 EP disclosed
US-5041460-A Antiallergens, antiinflammatory agents and leukotriene antagonists ICI AMERICAS INC. (US) 1991-08-20 US disclosed
EP-0337766-A1 Hetera-aliphatic carboxamides ICI AMERICAS INC. (US) 1989-10-18 EP disclosed