SCHEMBL9488902

SCHEMBL9488902

CC(C)(C)OC(=O)CC(O)c1c(CCCCCCCCc2ccccc2)ccc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
FAAH O00519 1/20 0.37
BACE1 P56817 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36
TRPA1 O75762 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GMNN O75496 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428159 0.80 CYSLTR2 (0.47) ADRB2ADRB1ADRB3FAAHTRPA1
SCHEMBL9560179 0.75 CYSLTR2 (0.56) ADRB2ADRB1ADRB3FAAH
SCHEMBL9561206 0.74 FAAH (0.37) ADRB2ADRB1ADRB3FAAHTRPA1
SCHEMBL27586622 0.71 MAPT (0.59) ADRB2ADRB1ADRB3FAAHMAPK1
SCHEMBL13356917 0.70 MMP2 (0.45)
SCHEMBL10578604 0.70 HDAC1 (0.56) ADRB2ADRB1ADRB3ALDH1A1HPGD
SCHEMBL9196120 0.69 MAPT (0.56) ADRB2ADRB1ADRB3FAAHMAPK1
SCHEMBL9485343 0.69 CYSLTR2 (0.49)
SCHEMBL5400156 0.69 GRIK1 (0.54)
SCHEMBL5400150 0.69 GRIK1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527175-A4 3-NAPHTHYL-3-CARBOXYALKYLTHIO OR OXY SUBSTITUTED ALKANOIC ACID LEUKOTRIENE ANTAGONISTS 1993-05-05 EP disclosed
EP-0527175-A1 3-NAPHTHYL-3-CARBOXYALKYLTHIO OR OXY SUBSTITUTED ALKANOIC ACID LEUKOTRIENE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1993-02-17 EP disclosed
WO-1991017149-A1 3-NAPHTHYL-3-CARBOXYALKYLTHIO OR OXY SUBSTITUTED ALKANOIC ACID LEUKOTRIENE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1991-11-14 WO disclosed