SCHEMBL9490484

SCHEMBL9490484

COc1cccc(C(C#N)(CCCNCCCc2ccccc2)C(C)C)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.57
CYP3A4 P08684 6/20 0.57
CYP3A5 P20815 1/20 0.57
SIGMAR1 Q99720 3/20 0.50
EBP Q15125 2/20 0.50
CACNA1B Q00975 3/20 0.44
HTR2A P28223 2/20 0.42
ABCC1 P33527 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
CHRM2 P08172 2/20 0.42
CYP2C19 P33261 2/20 0.42
ABCB11 O95342 2/20 0.42
KCNH2 Q12809 2/20 0.42
TSHR P16473 2/20 0.42
LMNA P02545 2/20 0.42
OPRM1 P35372 2/20 0.42
SLC22A1 O15245 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9492147 0.95 ABCB1 (0.60) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9492153 0.95 ABCB1 (0.60) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9491747 0.94 ABCB1 (0.57) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9490440 0.92 ABCB1 (0.57) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9490435 0.92 ABCB1 (0.57) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9492262 0.92 ABCB1 (0.56) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9492266 0.92 ABCB1 (0.56) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9492817 0.90 ABCB1 (0.57) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9490519 0.90 ABCB1 (0.57) ABCB1CYP3A4CYP3A5SIGMAR1EBP
SCHEMBL9639643 0.87 SIGMAR1 (0.64) ABCB1CYP3A4CYP3A5SIGMAR1EBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231003-B1 BASIC SUBSTITUTED PHENYLACETONITRILES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM BASF Aktiengesellschaft (DE) 1993-04-07 EP disclosed