SCHEMBL9639643

SCHEMBL9639643

CC(C)C(C#N)(CCCNCCCc1ccccc1)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.64
EBP Q15125 2/20 0.64
ABCB1 P08183 3/20 0.53
CYP3A4 P08684 2/20 0.53
CYP3A5 P20815 1/20 0.53
DRD2 P14416 1/20 0.50
DRD4 P21917 1/20 0.50
OPRM1 P35372 1/20 0.50
DRD3 P35462 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
KCNH2 Q12809 1/20 0.44
FDPS P14324 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9354199 0.95 SIGMAR1 (0.64) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9625375 0.95 SIGMAR1 (0.64) SIGMAR1EBPABCB1CYP3A4CYP3A5
Hydrochloric Acid SCHEMBL9357344 0.94 SIGMAR1 (0.62) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL10770803 0.92 SIGMAR1 (0.55) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9490838 0.92 SIGMAR1 (0.55) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9493520 0.89 SIGMAR1 (0.52) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9491747 0.87 ABCB1 (0.57) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9490484 0.87 ABCB1 (0.57) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9492266 0.86 ABCB1 (0.56) SIGMAR1EBPABCB1CYP3A4CYP3A5
SCHEMBL9492262 0.86 ABCB1 (0.56) SIGMAR1EBPABCB1CYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0270782-B1 THERAPEUTIC AGENTS FOR THE PROPHYLAXIS OF TUMOUR METASTASIS BASF Aktiengesellschaft (DE) 1992-08-12 EP disclosed
EP-0268100-B1 ACTIVE SUBSTANCES FOR USE IN THE TREATMENT OF TUMOURS BASF Aktiengesellschaft (DE) 1991-06-12 EP disclosed
EP-0270782-A2 Therapeutic agents for the prophylaxis of tumour metastasis BASF Aktiengesellschaft (DE) 1988-06-15 EP disclosed
EP-0268100-A1 Active substances for use in the treatment of tumours BASF Aktiengesellschaft (DE) 1988-05-25 EP disclosed