SCHEMBL949133

SCHEMBL949133

CN1CCn2c(cc3cc(O)ccc32)C1CC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 15/20 0.41
TSHR P16473 1/20 0.38
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
S1PR5 Q9H228 2/20 0.36
S1PR4 O95977 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945998 0.81 S1PR1 (0.54) S1PR1S1PR5S1PR4
SCHEMBL12320295 0.78 S1PR1 (0.54) S1PR1S1PR5S1PR4
SCHEMBL948546 0.75 S1PR1 (0.55) S1PR1S1PR5S1PR4
SCHEMBL949792 0.73 S1PR1 (0.34) S1PR1S1PR5S1PR4
SCHEMBL951026 0.71 S1PR1 (0.74) S1PR1S1PR5S1PR4
SCHEMBL948843 0.71 ESR2 (0.38) S1PR1OPRK1
SCHEMBL2446506 0.70 S1PR1 (0.46) S1PR1S1PR5S1PR4
SCHEMBL2446502 0.70 S1PR1 (0.46) S1PR1S1PR5S1PR4
SCHEMBL12320236 0.70 S1PR1 (0.46) S1PR1S1PR5S1PR4
SCHEMBL2017262 0.68 S1PR1 (0.53) S1PR1S1PR5S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed