SCHEMBL949792

SCHEMBL949792

CC(C)(C)OC(=O)CC1c2cc3cc(O)ccc3n2CCN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 13/20 0.34
ESR2 Q92731 1/20 0.33
MIF P14174 1/20 0.33
HTR6 P50406 1/20 0.32
S1PR4 O95977 1/20 0.32
S1PR5 Q9H228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL948843 0.92 ESR2 (0.38) S1PR1ESR2MIFHTR6
SCHEMBL14321088 0.81 S1PR1 (0.44) S1PR1S1PR4S1PR5
SCHEMBL2017781 0.81 S1PR1 (0.44) S1PR1S1PR4S1PR5
SCHEMBL946678 0.78 S1PR1 (0.45) S1PR1ESR2MIFHTR6
SCHEMBL948567 0.76 NR1H2 (0.32)
SCHEMBL948569 0.76 NR1H2 (0.32)
SCHEMBL949133 0.73 S1PR1 (0.41) S1PR1S1PR4S1PR5
SCHEMBL948764 0.69 S1PR1 (0.63) S1PR1S1PR4S1PR5
SCHEMBL2446502 0.69 S1PR1 (0.46) S1PR1MIFS1PR4S1PR5
SCHEMBL2446506 0.69 S1PR1 (0.46) S1PR1MIFS1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed