SCHEMBL948843

SCHEMBL948843

CC(C)(C)OC(=O)CC1c2cc3cc(O)ccc3n2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.38
HTR6 P50406 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NR1H2 P55055 7/20 0.33
NR1H3 Q13133 5/20 0.33
MIF P14174 1/20 0.33
S1PR1 P21453 2/20 0.33
TGFBR1 P36897 1/20 0.33
GPR119 Q8TDV5 1/20 0.32
RXRA P19793 2/20 0.32
PIK3CD O00329 1/20 0.32
OPRK1 P41145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949792 0.92 S1PR1 (0.34) ESR2HTR6MIFS1PR1
SCHEMBL948567 0.84 NR1H2 (0.32) MEN1KMT2ANR1H2NR1H3GPR119
SCHEMBL948569 0.84 NR1H2 (0.32) MEN1KMT2ANR1H2NR1H3GPR119
SCHEMBL14321088 0.81 S1PR1 (0.44) S1PR1
SCHEMBL2017781 0.81 S1PR1 (0.44) S1PR1
SCHEMBL946678 0.78 S1PR1 (0.45) ESR2HTR6MIFS1PR1
SCHEMBL948764 0.76 S1PR1 (0.63) S1PR1
SCHEMBL947762 0.75 S1PR1 (0.64) S1PR1
SCHEMBL949133 0.71 S1PR1 (0.41) S1PR1OPRK1
SCHEMBL2446502 0.69 S1PR1 (0.46) MIFS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005295-A1 MODULATORS OF THE SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed