SCHEMBL9492425

SCHEMBL9492425

COc1cc(CCN(C)CCCC(C#N)(c2ccccc2)c2cc(OC)cc(OC)c2)cc(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EBP Q15125 3/20 0.50
SIGMAR1 Q99720 3/20 0.50
DRD2 P14416 4/20 0.47
DRD3 P35462 4/20 0.47
OPRM1 P35372 3/20 0.47
CYP2D6 P10635 2/20 0.47
DRD4 P21917 2/20 0.47
ABCB1 P08183 6/20 0.44
CYP3A4 P08684 5/20 0.44
ABCC1 P33527 4/20 0.44
KCNH2 Q12809 4/20 0.44
TSHR P16473 3/20 0.44
LMNA P02545 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP2C19 P33261 2/20 0.44
ABCB11 O95342 2/20 0.44
CACNA1F O60840 2/20 0.44
HTR1A P08908 2/20 0.44
ADRA2A P08913 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493593 0.98 SIGMAR1 (0.52) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL9490822 0.89 SIGMAR1 (0.53) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL10453764 0.83 SIGMAR1 (0.54) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL11820903 0.82 CYP3A4 (0.64) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL9492427 0.81 DRD2 (0.50) SIGMAR1DRD2DRD3OPRM1CYP2D6
SCHEMBL10453936 0.79 ABCB1 (0.40) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL9490429 0.79 SIGMAR1 (0.63) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL10452583 0.79 SIGMAR1 (0.63) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL9492261 0.78 SIGMAR1 (0.76) EBPSIGMAR1DRD2DRD3OPRM1
SCHEMBL10452662 0.78 SIGMAR1 (0.76) EBPSIGMAR1DRD2DRD3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231003-B1 BASIC SUBSTITUTED PHENYLACETONITRILES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM BASF Aktiengesellschaft (DE) 1993-04-07 EP disclosed
US-4968717-A SEROTONIN-AND CALCIUM-ANTAGONISTS BASF AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed