SCHEMBL9494064

SCHEMBL9494064

FC(F)(F)c1cc(Cl)c2cccc(C(Cl)Cl)c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.43
ADORA2A P29274 6/20 0.38
ADORA1 P30542 6/20 0.38
LMNA P02545 2/20 0.38
KCNH2 Q12809 7/20 0.37
CYP3A4 P08684 3/20 0.37
ADORA3 P0DMS8 2/20 0.37
CYP2D6 P10635 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ADORA2B P29275 1/20 0.37
CYP2C19 P33261 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
NR1I2 O75469 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
HTR1A P08908 1/20 0.37
TSHR P16473 1/20 0.37
CNR1 P21554 1/20 0.37
GLRA1 P23415 1/20 0.37
SLC6A2 P23975 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9493850 0.88 LMNA (0.38) NT5ELMNACYP3A4KDM4ENR1I2
SCHEMBL2710931 0.82 NT5E (0.48) NT5ELMNAKDM4ECYP2C19CYP1A2
SCHEMBL1258312 0.79 KCNH2 (0.47) NT5EADORA2AADORA1LMNAKCNH2
SCHEMBL2711028 0.79 NT5E (0.49) NT5EADORA2AADORA1LMNACYP3A4
SCHEMBL3628877 0.78 NT5E (0.44) NT5EADORA2AADORA1LMNAKCNH2
SCHEMBL3628880 0.78 NT5E (0.44) NT5EADORA2AADORA1LMNAKCNH2
SCHEMBL3631708 0.78 ENPP1 (0.56) NT5EADORA2AADORA1LMNAKDM4E
SCHEMBL2711191 0.78 ELANE (0.48) NT5ELMNAKDM4ETP53HTT
SCHEMBL9493205 0.76 NT5E (0.43) NT5EADORA2AADORA1LMNAKDM4E
SCHEMBL9493460 0.76 NT5E (0.43) NT5EADORA2AADORA1LMNAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0113432-B1 CHLOROMETHYL QUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE ALKALOIDA VEGYéSZETI GYáR (HU) 1993-03-17 EP claimed
EP-0113432-A1 Chloromethyl quinoline derivatives, process for their preparation and their use ALKALOIDA VEGYéSZETI GYáR (HU) 1984-07-18 EP claimed