SCHEMBL9497011

SCHEMBL9497011

CCCCCOc1ccc(C#Cc2ccc(C)cn2)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GRM5 P41594 1/20 0.34
S1PR4 O95977 1/20 0.32
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
S1PR5 Q9H228 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9496170 0.96 GRM5 (0.35) ALDH1A1HPGDGAAMAPTTHRB
SCHEMBL9498411 0.93 GRM5 (0.36) ALDH1A1GAAMAPTGRM5
SCHEMBL9497092 0.89 GRM5 (0.38) GRM5
SCHEMBL9497884 0.87 ALDH1A1 (0.34) ALDH1A1HPGDMAPTS1PR1S1PR3
SCHEMBL9496652 0.86 RAB9A (0.40) ALDH1A1HPGDMAPTNPSR1S1PR1
SCHEMBL9498182 0.86 RAB9A (0.38) ALDH1A1HPGDMAPTS1PR1S1PR3
SCHEMBL9496009 0.86 RAB9A (0.43) ALDH1A1HPGDGAAMAPTTHRB
SCHEMBL9496316 0.85 RAB9A (0.42) ALDH1A1HPGDGAAMAPTNPSR1
SCHEMBL10511057 0.85 RAB9A (0.42) ALDH1A1HPGDGAAMAPTNPSR1
SCHEMBL9497274 0.85 RAB9A (0.42) ALDH1A1HPGDGAAMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0306505-B1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1993-03-24 EP disclosed
US-5068053-A Liquid crystals for optical apparatus MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-11-26 US disclosed
EP-0306505-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007523-A1 ACETYLENE DERIVATIVES AS COMPONENTS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed