SCHEMBL9501126

SCHEMBL9501126

O=C(O)Oc1cn(C2CC2)c2cc(N3CCNCC3)c(F)c(F)c2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.56
ALDH1A1 P00352 6/20 0.56
HPGD P15428 5/20 0.56
HSD17B10 Q99714 5/20 0.56
LMNA P02545 4/20 0.56
CYP1A2 P05177 1/20 0.56
TOP2A P11388 1/20 0.56
CYP2C9 P11712 1/20 0.56
TOP2B Q02880 1/20 0.56
KCNH2 Q12809 2/20 0.50
HRH3 Q9Y5N1 1/20 0.50
MAPT P10636 1/20 0.40
BRD4 O60885 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
CYP2J2 P51589 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 1/20 0.39
CASP3 P42574 1/20 0.39
CASP9 P55211 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9049511 0.91 KCNH2 (0.59) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9501385 0.91 KDM4E (0.53) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9502081 0.88 KCNH2 (0.66) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL10683412 0.85 KCNH2 (0.47) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9502044 0.85 KCNH2 (0.52) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9501123 0.84 KDM4E (0.70) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL1857925 0.84 KDM4E (0.76) KDM4EALDH1A1HPGDHSD17B10LMNA
Hydrochloric Acid SCHEMBL9808640 0.83 KDM4E (0.74) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL1858180 0.82 KCNH2 (0.76) KDM4EALDH1A1HPGDHSD17B10LMNA
SCHEMBL9503656 0.81 KCNH2 (0.62) KDM4EALDH1A1HPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312085-B1 NOVEL QUINOLINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND ANTIBACTERIAL AGENT CONTAINING THEM Dainippon Pharmaceutical Co., Ltd. (JP) 1993-05-12 EP claimed