SCHEMBL9502081

SCHEMBL9502081

CC1CN(c2cc3c(c(F)c2F)c(=O)c(OC(=O)O)cn3C2CC2)CCN1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.66
HRH3 Q9Y5N1 1/20 0.66
KDM4E B2RXH2 7/20 0.47
ALDH1A1 P00352 7/20 0.47
HPGD P15428 6/20 0.47
HSD17B10 Q99714 6/20 0.47
POLB P06746 2/20 0.47
PRKD3 O94806 1/20 0.47
ALOX15 P16050 1/20 0.47
OPRM1 P35372 1/20 0.47
CLK2 P49760 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.43
TOP2A P11388 1/20 0.43
CYP2C9 P11712 1/20 0.43
TOP2B Q02880 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1858180 0.94 KCNH2 (0.76) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9503656 0.93 KCNH2 (0.62) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9502044 0.89 KCNH2 (0.52) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9501126 0.88 KDM4E (0.56) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL10808537 0.86 KDM4E (0.59) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9501145 0.85 KCNH2 (0.87) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL10683412 0.85 KCNH2 (0.47) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9500961 0.83 KCNH2 (0.52) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9435843 0.83 MEN1 (0.57) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL9049511 0.82 KCNH2 (0.59) KCNH2HRH3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312085-B1 NOVEL QUINOLINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND ANTIBACTERIAL AGENT CONTAINING THEM Dainippon Pharmaceutical Co., Ltd. (JP) 1993-05-12 EP claimed